GSK Kinase Inhibitor 1

This collection of 367 kinase inhibitors was provided by GlaxoSmithKline (GSK) in February 2012. Together, the inhibitors span 30 chemotypes that have been published by GSK in peer-reviewed scientific journals. The GSK collection is currently available to Harvard and Dana-Farber Cancer Institute investigators under a Material Transfer Agreement, a primary requirement of which is that results obtained from screening this collection must be placed in the public domain via PubChem BioAssay.

Number of Compounds 367
Plate Numbers 3303-3304 (2 Plates)
Concentration Information 3.3 mM in DMSO

This library was retired in July 2017.  It is now available through the University of North Carolina as the UNC SGC Published Kinase Inhibitor Set. If you're interested in screening the UNC library, follow the instructions on the linked pages to get access. Here is a link to the required MTA  to be filled out by each investigator interested in screening the library.  

384-well Plate Format

 A signed MTA and permission is required to screen this library; ICCB-L screeners interested should contact Jennifer Smith for more details.